DS43260857
Product Specifications
CAS Number
1612158-07-2
Target
Sodium Channel
Related Pathways
Membrane transporter/Ion channel
Bioactivity
DS43260857 is a potent NaV1.7 inhibitor with high inhibitory effects on both human and mouse NaV1.7, exhibiting IC50 values of 6.6 μM for hNaV1.1, 14 μM for hNaV1.5, 0.015 μM for hNaV1.7, and 0.061 μM for mNaV1.7 [1].
Smiles
CC=1C=2C(N(C1)C=3C=C(C(F)(F)F)C=NC3)=CC=C(C(NS(=O)(=O)C4CC4)=O)C2
Molecular Formula
C19H16F3N3O3S
Molecular Weight
423.41
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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