CSF1R-IN-23
Product Specifications
CAS Number
2935480-17-2
Target
C-Fms
Related Pathways
Tyrosine Kinase/Adaptors
Bioactivity
CSF1R-IN-23 (Compound 7dri), a selective colony-stimulating factor-1 receptor (CSF1R) inhibitor, exhibits an IC50 of 36.1 nM. This compound acts as an antineuroinflammatory agent in a mouse model and is noted for its blood-brain barrier (BBB) permeability [1].
Smiles
N(C(=O)C1=NOC(C)=C1)C2=C(C=C(C=C2)C3CC(C)(C)NC(C)(C)C3)C=4CCC(C)CC4
Molecular Formula
C27H37N3O2
Molecular Weight
435.6
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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