Salvinorin A Carbamate
Product Specifications
CAS Number
858345-57-0
Target
Others, Opioid Receptor
Related Pathways
Endocrinology/Hormones, GPCR/G Protein, Others, Neuroscience
Bioactivity
Salvinorin A carbamate, a potent κ-opioid receptor (KOR) full agonist, exhibits nearly the same potency as salvinorin A, with EC50 values of 6.2 and 4.5 nM, respectively, for activating the human KOR to augment the binding of [35S]GTPγS. Enhancing biological stability, the addition of a carbamate group to salvinorin A reduces deacetylation.
Smiles
COC(=O)[C@@H]1C[C@H](OC(N)=O)C(=O)[C@H]2[C@@]1(C)CC[C@H]1C(=O)O[C@@H](C[C@]21C)c1ccoc1
Molecular Formula
C22H27NO8
Molecular Weight
433.457
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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