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M084 hydrochloride

Product Specifications

CAS Number

1992047-63-8

Target

Others, TRP/TRPV Channel

Related Pathways

Others, Membrane transporter/Ion channel

Bioactivity

M084 hydrochloride, a TRPC4/5 channel blocker, exhibits IC50 values of 10.3 μM and 8.2 μM, respectively. This compound is noted for its antidepressant and anxiolytic effects [1] [2].

Smiles

N(CCCC)C=1NC=2C(N1)=CC=CC2.Cl

Molecular Formula

C11H16ClN3

Molecular Weight

225.72

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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