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CGP36216 hydrochloride

Product Specifications

CAS Number

1781834-71-6

Target

Others, GABA Receptor

Related Pathways

Neuroscience, Membrane transporter/Ion channel, Others

Bioactivity

CGP36216 hydrochloride acts as a selective antagonist at the presynaptic GABA receptor, specifically binding to the GABAB receptor with a Ki value of 0.3 μM. This compound is leveraged in research focused on anxiety and trauma-related disorders [1] [2].

Smiles

P(CCCN)(CC)(=O)O.Cl

Molecular Formula

C5H15ClNO2P

Molecular Weight

187.6

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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