DB21, Galectin-1 Antagonist

Product Specifications

CAS Number

1623027-80-4

Target

Galectin

Related Pathways

Immunology/Inflammation

Bioactivity

DB21, Galectin-1 Antagonist, is a peptidomimetic conjugated with dibenzofuran, serving as an allosteric inhibitor of galectin-1 (GAL1) interactions with glycans on cell surfaces. This compound enhances the inhibition of angiogenesis and tumor growth in melanoma, lung adenocarcinoma, and ovarian cancer models [1].

Smiles

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