GK718
Product Specifications
Target
HDAC
Related Pathways
DNA Damage/DNA Repair, Chromatin/Epigenetic
Bioactivity
GK718, a selective HDAC1/3 inhibitor with IC50 values of 259 nM and 139 nM, respectively, elevates acetylated histone H3 levels in cells and mitigates Bleomycin-induced pulmonary fibrosis in mice [1].
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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