What is the catalog number for PNMT-IN-1?

The catalog number for PNMT-IN-1 is T81432.

What sizes are available for PNMT-IN-1?

PNMT-IN-1 is available in the following size(s): 5 mg, 50 mg.

How many pack sizes does PNMT-IN-1 come in?

PNMT-IN-1 is available in 2 different pack sizes.

Is PNMT-IN-1 in stock?

PNMT-IN-1 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures PNMT-IN-1?

PNMT-IN-1 is manufactured by Molfinity.

What is the estimated delivery time for PNMT-IN-1?

Estimated delivery time for PNMT-IN-1 is approximately 10 business day(s), depending on your location.

PNMT-IN-1

Product Specifications

Target

Adrenergic Receptor, Others

Related Pathways

Neuroscience, GPCR/G Protein, Others

Bioactivity

PNMT-IN-1 (inhibitor 4) is a selective second generation inhibitor [1] of phenylethanolamine N-methyltransferase (PNMT), exhibiting a Ki value of 1.2 nM and an IC50 value of 81 nM. Additionally, it disrupts the activity of DNMT1 and DNMT3b, with IC50 values of 61 μM and 17 μM, respectively, and antagonizes the action of epinephrine.