TRPV2-selective blocker 1
Product Specifications
CAS Number
2242724-49-6
Target
TRP/TRPV Channel, Others
Related Pathways
Others, Membrane transporter/Ion channel
Bioactivity
TRPV2-selective blocker 1 (compound IV2-1) is a selective inhibitor of the TRPV2 channel, with an IC50 value of 6.3 μM, specifically targeting the TRPV2 channel without affecting TRPV1, TRPV3, or TRPV4 channels, and effectively suppresses TRPV2-mediated calcium influx in macrophages, inhibiting their phagocytic activity [1].
Smiles
O=C(C)CC(C(=C1SCCS1)C=2C=CC=CC2)C
Molecular Formula
C15H18OS2
Molecular Weight
278.43
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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