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Jingzhaotoxin XI

Product Specifications

Target

Sodium Channel

Related Pathways

Membrane transporter/Ion channel

Bioactivity

Jingzhaotoxin XI (JZTX-XI) is a potent inhibitor of sodium conductance with an IC50 of 124 nM, and it significantly delays the rapid inactivation of Na_v1.5, with an EC50 of 1.18±0.2 μM, when expressed in Chinese hamster ovary (CHO-K1) cells [1].

Molecular Formula

C158H234N44O47S7

Molecular Weight

3726.27

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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