ω-Conotoxin CVIB

Product Specifications

CAS Number

325164-09-8

Target

Sodium Channel

Related Pathways

Membrane transporter/Ion channel

Bioactivity

?-Conotoxin CVIB is an antagonist of non-selective N- and P/Q-type voltage-gated calcium channels (VGCCs) . It inhibits depolarization-activated whole-cell VGCC currents in dorsal root ganglion (DRG) neurons, exhibiting a pIC50 of 7.64 [1].

Smiles

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