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FPR1 antagonist 2

Product Specifications

Target

Apoptosis|||Others

Related Pathways

Others|||Apoptosis

Bioactivity

Compound 25b, an FPR1 antagonist, exhibits potent inhibition of the formyl peptide receptor 1 with an IC50 of 70 nM. It concurrently hampers cell proliferation and triggers apoptosis, diminishing cell growth and migration, yet paradoxically augments angiogenesis [1].

Molecular Formula

C25H25F3O5

Molecular Weight

462.46

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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