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FD2157

Product Specifications

Target

PI3K|||Apoptosis

Related Pathways

PI3K/Akt/mTOR signaling|||Apoptosis

Bioactivity

FD2157, a photosensitive PI3K inhibitor, exhibits inhibitory IC50 values of 43 nM for PI3K?, 83 nM for PI3K?, 84 nM for PI3K?, and 14 nM for PI3K?. Upon exposure to 365 nm UV light, FD2157 effectively inhibits cancer cell proliferation and induces apoptosis [1].

Molecular Formula

C27H21ClN6O8S

Molecular Weight

625.01

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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