FD2157
Product Specifications
Target
PI3K|||Apoptosis
Related Pathways
PI3K/Akt/mTOR signaling|||Apoptosis
Bioactivity
FD2157, a photosensitive PI3K inhibitor, exhibits inhibitory IC50 values of 43 nM for PI3K?, 83 nM for PI3K?, 84 nM for PI3K?, and 14 nM for PI3K?. Upon exposure to 365 nm UV light, FD2157 effectively inhibits cancer cell proliferation and induces apoptosis [1].
Molecular Formula
C27H21ClN6O8S
Molecular Weight
625.01
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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