PKM2-IN-4
Product Specifications
Target
Others, PKM
Related Pathways
Others, Metabolism
Bioactivity
Compound 5C, referred to as Pkm2-in-4, is a selective PKM2 inhibitor (IC50 = 0.35 μM) that modulates pyruvate-dependent respiration and promotes mitochondrial H2O2 production rate and electron transport system coupling [1].
Molecular Formula
C15H17BrClNO3Se
Molecular Weight
453.62
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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