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M3/PDE4 modulator-1

Product Specifications

Target

AChR|||Others|||PDE

Related Pathways

Neuroscience|||Others|||Metabolism

Bioactivity

M3/PDE4 Modulator-1 (compound 10f) serves as a bifunctional entity functioning both as an M3 mAChR antagonist and a PDE4 inhibitor. When administered intravenously at concentrations ranging from 10 to 1000 nM/kg, this compound effectively diminishes eosinophil influx into cysts within the OVA rat model [1].

Molecular Formula

C38H41Cl2N3O8S

Molecular Weight

770.72

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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