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BET-IN-17

Product Specifications

Target

Epigenetic Reader Domain

Related Pathways

Chromatin/Epigenetic

Bioactivity

BET-IN-17, also known as compound 16, serves as a pan-inhibitor for BET, exhibiting inhibitory potencies (pIC50) of 7.8 for BET BD1 and 7.6 for BET BD2 [1].

Molecular Formula

C30H36N4O2

Molecular Weight

484.63

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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