ET receptor antagonist 2
Product Specifications
Target
Estrogen Receptor/ERR
Related Pathways
Endocrinology/Hormones
Bioactivity
ET Receptor Antagonist 2 (Compound 16j) is an orally active ET receptor antagonist with an IC50 of 0.22 nM, suitable for pulmonary arterial hypertension (PAH) research. It has been shown to mitigate monocrotaline-induced PAH in a rat model [1].
Molecular Formula
C22H25N5O5S
Molecular Weight
471.53
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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