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JNK-1-IN-2

Product Specifications

Target

JNK

Related Pathways

MAPK

Bioactivity

"JNK-1-IN-2 (Compound c6) is a potent inhibitor of JNK-1 with an IC50 of 33.5 nM, and also exhibits inhibitory effects on JNK-2 and JNK-3 with IC50 values of 112.9 nM and 33.2 nM, respectively. This compound effectively inhibits the phosphorylation of c-Jun and has shown potential in reversing lung impairment, making it relevant for research into pulmonary fibrosis [1]."

Molecular Formula

C16H20BrN5O

Molecular Weight

378.27

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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