Anticancer agent 135
Product Specifications
Target
Androgen Receptor
Related Pathways
Endocrinology/Hormones
Bioactivity
Anticancer agent 135 (compound 26h) is a potent androgen receptor (AR) antagonist that blocks AR nuclear translocation and inhibits AR/AR-V7 heterodimerization to suppress downstream gene transcription, demonstrating strong efficacy in prostate cancer xenograft models [1].
Molecular Formula
C23H21F3N4OS
Molecular Weight
458.5
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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