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KV1.3-IN-1

Product Specifications

Target

Potassium Channel

Related Pathways

Membrane transporter/Ion channel

Bioactivity

KV1.3-IN-1 (Compound trans-18) is a selective KV1.3 channel inhibitor with IC50 values of 230 nM in Ltk cells and 26.12 nM in PHA-activated T-lymphocytes, disrupting intracellular Ca2+ signaling and impeding T-cell activation, proliferation, and colony formation [1].

Molecular Formula

C23H30N2O4S

Molecular Weight

430.56

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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