TGR5 agonist 3

2148317-51-3

Others|||GPCR19

Others|||GPCR/G Protein

Compound 8, a cholic acid derivative, functions as a selective TGR5 agonist and exhibits an EC50 value of 5 ?M [1].

C(CCC)[C@]1(O)[C@@]2([C@@]([C@]3(C)[C@](C1)(C[C@H](O)CC3)[H])(C[C@H](O)[C@@]4(C)[C@]2(CC[C@@]4([C@@H](CCC(O)=O)C)[H])[H])[H])[H]

C28H48O5

464.68

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