A3AR agonist 2
Product Specifications
Target
Adenosine Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Bioactivity
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM. This compound is utilized in research pertaining to inflammatory diseases, ischemia, cancer, neuropathic pain, liver diseases, and other chronic conditions [1].
Molecular Formula
C34H34N6O6
Molecular Weight
622.67
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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