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A3AR agonist 2

Product Specifications

Target

Adenosine Receptor

Related Pathways

Neuroscience, GPCR/G Protein

Bioactivity

Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM. This compound is utilized in research pertaining to inflammatory diseases, ischemia, cancer, neuropathic pain, liver diseases, and other chronic conditions [1].

Molecular Formula

C34H34N6O6

Molecular Weight

622.67

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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