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BMPR2-IN-1

Product Specifications

Target

TGF-beta/Smad|||Others

Related Pathways

Stem Cells|||Others

Bioactivity

BMPR2-IN-1 (Compound 8a), is a potent inhibitor of BMPR2, exhibiting an IC50 value of 506 nM and a Kd of 83.5 nM. It is utilized in the study of various diseases including pulmonary arterial hypertension, Alzheimer's disease, and cancer [1].

Smiles

O=C1C2=CC(NC3=CC=NC(NC4=CC=C(CCN1)C=C4)=N3)=NN2

Molecular Formula

C16H15N7O

Molecular Weight

321.34

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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