CaSR antagonist-1
Product Specifications
CAS Number
1219811-83-2
Target
CaSR
Related Pathways
GPCR/G Protein
Bioactivity
CaSR Antagonist-1 is a potent inhibitor of the calcium-sensing receptor (CaSR) with an inhibitory concentration (IC50) of 50 nM, suitable for the investigation of diseases related to dysregulated bone or mineral homeostasis, including osteoporosis [1].
Smiles
C(CC1=CC=CC=C1)N2C(=NC(C)=C(C2=O)C3=CC(=C(C)S3)C4=CC=CC=N4)C5=C(O)C(F)=CC=C5
Molecular Formula
C29H24FN3O2S
Molecular Weight
497.58
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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