BET-IN-16
Product Specifications
CAS Number
2089390-09-8
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Bioactivity
BET-IN-16 (Comp I), a bromodomain and extra-terminal (BET) inhibitor, demonstrates anticancer activity by impeding the growth of prostate cancer cells. It exhibits potent inhibitory effects with half-maximal inhibitory concentration (IC50) values of 0.043 μM for LNCaP cells and 0.034 μM for 22Rv1 cells [1].
Smiles
C(C)(N1C=2C(C(=C1)C3=CC=C(C(O)=O)C=C3)=NC=C(C2)C=4C(C)=NOC4C)(C5=CC=CC=N5)C6=CC=CC=N6
Molecular Formula
C31H25N5O3
Molecular Weight
515.56
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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