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PROTAC BRD3/BRD4-L degrader-2

Product Specifications

Target

Epigenetic Reader Domain|||PROTACs

Related Pathways

Chromatin/Epigenetic|||PROTAC

Bioactivity

PROTAC BRD3/BRD4-L degrader-2, a PROTAC molecule, selectively degrades cellular BRD3 and BRD4-L with K i values of 16.91 and 2.8 nM, respectively, and exhibits robust antitumor activity in mouse xenograft models, serving as a research tool for cancer [1].

Molecular Formula

C43H44ClN7O3

Molecular Weight

742.31

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Product Datasheet

https://www.targetmol.com/attachment/DataSheet/123792051979419654/T78956

Available Sizes

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