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HNTS1R agonist-1

Product Specifications

Target

Neurotensin Receptor

Related Pathways

GPCR/G Protein

Bioactivity

Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (BBB) . It not only enhances motor function but also improves memory in a mouse model of Parkinson's disease (PD) . Additionally, this compound is an analog of Neurotensin (8-13) and demonstrates neuroprotective properties [1].

Molecular Formula

C37H62N10O9

Molecular Weight

790.95

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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