WCA-814
Product Specifications
Target
Androgen Receptor
Related Pathways
Endocrinology/Hormones
Bioactivity
WCA-814, an androgen receptor (AR) antagonist-Hsp90 inhibitor conjugate, induces degradation of both full-length and AR-V7, exhibiting cytotoxic effects in prostatic cancer cells with half maximal inhibitory concentrations (IC50) of 171.2 nM and 26.5 nM for LNCaP and 22Rv1 cells, respectively [1].
Molecular Formula
C46H53ClN10O5
Molecular Weight
861.43
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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