EGFR-IN-78
Product Specifications
Target
Apoptosis|||EGFR
Related Pathways
Apoptosis|||Angiogenesis|||JAK/STAT signaling|||Tyrosine Kinase/Adaptors
Bioactivity
EGFR-IN-78 (compound A5), a 2-aminopyrimidine derivative, serves as a reversible EGFR C797S-TK inhibitor and an apoptosis inducer. It exhibits anti-proliferative properties, impedes EGFR phosphorylation, and induces G2/M phase cell cycle arrest [1].
Molecular Formula
C23H32BrN7O2S
Molecular Weight
550.51
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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