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CDK2/Bcl2-IN-1

Product Specifications

Target

CDK

Related Pathways

Cell Cycle/Checkpoint

Bioactivity

CDK2/Bcl2-IN-1 (compound 1) is a saponin-based inhibitor of CDK-2 (IC50=117.6 nM) with potent cytotoxic effects on cancer cells, also inhibiting Bcl-2 and promoting apoptosis in A549 lung cancer cells [1].

Molecular Formula

C35H56O10S

Molecular Weight

668.88

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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