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D3R/MOR antagonist 2

Product Specifications

Target

Dopamine Receptor, Opioid Receptor

Related Pathways

Neuroscience, Endocrinology/Hormones, GPCR/G Protein

Bioactivity

Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR partial agonism and may reduce opioid-misuse liability through D3R antagonism [1].

Molecular Formula

C25H31ClN2O

Molecular Weight

410.98

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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