D3R/MOR antagonist 2
Product Specifications
Target
Dopamine Receptor, Opioid Receptor
Related Pathways
Neuroscience, Endocrinology/Hormones, GPCR/G Protein
Bioactivity
Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR partial agonism and may reduce opioid-misuse liability through D3R antagonism [1].
Molecular Formula
C25H31ClN2O
Molecular Weight
410.98
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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