DiPT-4
Product Specifications
Target
Topoisomerase, Apoptosis, PARP
Related Pathways
Apoptosis, Chromatin/Epigenetic, DNA Damage/DNA Repair
Bioactivity
DiPT-4, a dual TOP1/PARP1 inhibitor, effectively induces DNA double-strand breaks (DSBs), cell cycle arrest, and apoptosis in cancer cells, with potential to circumvent drug resistance [1].
Molecular Formula
C32H22FN5O4S
Molecular Weight
591.61
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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