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DiPT-4

Product Specifications

Target

Topoisomerase, Apoptosis, PARP

Related Pathways

Apoptosis, Chromatin/Epigenetic, DNA Damage/DNA Repair

Bioactivity

DiPT-4, a dual TOP1/PARP1 inhibitor, effectively induces DNA double-strand breaks (DSBs), cell cycle arrest, and apoptosis in cancer cells, with potential to circumvent drug resistance [1].

Molecular Formula

C32H22FN5O4S

Molecular Weight

591.61

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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