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A011

Product Specifications

Target

ATM/ATR|||Apoptosis

Related Pathways

Apoptosis|||DNA Damage/DNA Repair|||PI3K/Akt/mTOR signaling

Bioactivity

A011, a potent and selective ataxia-telangiectasia mutated (ATM) inhibitor, exhibits an IC50 of 1.0 nM and triggers apoptosis as well as G2/M phase cell cycle arrest when combined with CPT-11, displaying notable antitumor activity [1].

Molecular Formula

C27H28N6O

Molecular Weight

452.55

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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