SJ1461
Product Specifications
CAS Number
2924546-70-1
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Bioactivity
SJ1461 is a potent, orally active inhibitor of the BET family, selectively targeting and inhibiting BRD2 (BD1), BRD2 (BD2), BRD4 (BD1), and BRD4 (BD2) with respective IC50 values of 1.6 nM, 0.1 nM, 6.5 nM, and 0.2 nM [1].
Smiles
CC=1C2=C(N3C([C@H](CC(NC4=NN=CS4)=O)N=C2C5=CC=C(Cl)C=C5)=NN=C3C)SC1C
Molecular Formula
C21H18ClN7OS2
Molecular Weight
484
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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