What is the catalog number for ERK1/2 inhibitor 9?

The catalog number for ERK1/2 inhibitor 9 is T78190.

What sizes are available for ERK1/2 inhibitor 9?

ERK1/2 inhibitor 9 is available in the following size(s): 5 mg, 50 mg.

How many pack sizes does ERK1/2 inhibitor 9 come in?

ERK1/2 inhibitor 9 is available in 2 different pack sizes.

Is ERK1/2 inhibitor 9 in stock?

ERK1/2 inhibitor 9 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures ERK1/2 inhibitor 9?

ERK1/2 inhibitor 9 is manufactured by Molfinity.

What is the estimated delivery time for ERK1/2 inhibitor 9?

Estimated delivery time for ERK1/2 inhibitor 9 is approximately 10 business day(s), depending on your location.

ERK1/2 inhibitor 9

Product Specifications

CAS Number

2169302-75-2

Target

ERK

Related Pathways

MAPK

Bioactivity

ERK1/2 Inhibitor 9 (Probe 1), a covalent antagonist of ERK1/2, exhibits sub-micromolar efficacy in cellular assays (A375 GI50=0.47 μM) and facilitates the reduction of phospho-ERK1/2 levels. When conjugated with trans-cyclo-octene (TCO) and Tz-Thalidomide (tetrazine-tagged Thalidomide), it forms the corresponding ERK-CLIPTAC, promoting targeted ERK1/2 degradation [1].