CS640
Product Specifications
CAS Number
2388506-83-8
Target
Others
Related Pathways
Others
Bioactivity
CS640 is a selective calmodulin-dependent kinase inhibitor, targeting multiple isoforms, namely CaMK1D, CaMK1B, CaMK1A, CaMK1G, PIP5K1C, MEK5, RIPK4, and MLK3, with respective IC50 values of 0.08, 0.03, 0.001, 0.001, 11.2, 0.025, 5.69, and 2.75 μM. Additionally, CS640 exhibits inhibitory properties toward CYP450 enzymes 2C9 and 2C19 with IC50 values of 6 and 10 μM, correspondingly [1].
Smiles
N(C=1C(C(N)=O)=CN=C(N1)N2C[C@@H](N)CCC2)C=3C=C(C(C)C)N=C(C(C)C)C3
Molecular Formula
C21H31N7O
Molecular Weight
397.52
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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