HIF-1α-IN-2 hydrochloride
Product Specifications
Target
HIF/HIF Prolyl-Hydroxylase
Related Pathways
Metabolism, Chromatin/Epigenetic
Bioactivity
HIF-1α-IN-2 hydrochloride is a potent HIF-1α inhibitor exhibiting anticancer activity, with IC50 values of 28 nM in MDA-MB-231 cells and 15 nM in MiaPaCa-2 cells, effectively suppressing HIF-1α expression by inhibiting transcription and protein translation [1].
Molecular Formula
C21H20ClN3OS
Molecular Weight
397.92
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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