Fosnetupitant chloride monohydrochloride
Product Specifications
CAS Number
1643757-72-5
Target
Neurokinin receptor
Related Pathways
GPCR/G Protein, Neuroscience
Bioactivity
Fosnetupitant chloride monohydrochloride (Pro-netupitant chloride monohydrochloride) is a selective NK1 antagonist exhibiting high affinity for the human NK1 receptor with a pK i value of 9.5, and a lower affinity for the NK3 receptor with a pK i of 6.1. It serves as a methylene phosphate prodrug of Netupitant [1].
Smiles
O=C(C(C)(C)C1=CC(C(F)(F)F)=CC(C(F)(F)F)=C1)N(C)C2=CN=C(N3CC[N+](COP(O)(O)=O)(CC3)C)C=C2C4=C(C)C=CC=C4.[Cl-].Cl
Molecular Formula
C31H37Cl2F6N4O5P
Molecular Weight
761.52
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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