PROTAC BCR-ABL Degrader-1
Product Specifications
Target
Bcr-Abl, PROTACs
Related Pathways
Tyrosine Kinase/Adaptors, PROTAC, Cytoskeletal Signaling, Angiogenesis
Bioactivity
PROTAC BCR-ABL Degrader-1 (compound PROTAC 1), featuring a 2-oxoethyl linker, induces Bcr-Abl degradation via the ubiquitin-proteasome pathway and exhibits antiproliferative effects on K562 cells, indicating its potential in cancer research [1].
Molecular Formula
C43H40N10O6
Molecular Weight
792.84
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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