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SIAIS100 TFA

Product Specifications

Target

PROTACs, Bcr-Abl

Related Pathways

PROTAC, Tyrosine Kinase/Adaptors, Angiogenesis, Cytoskeletal Signaling

Bioactivity

SIAIS100 TFA is a potent BCR-ABL PROTAC degrader with a DC50 of 2.7 nM, used in chronic myeloid leukemia (CML) research [1].

Molecular Formula

C46H51ClF5N9O7S

Molecular Weight

1004.46

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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