MY-1076
Product Specifications
CAS Number
3008262-76-5
Target
Apoptosis, YAP
Related Pathways
Apoptosis, Stem Cells
Purity
0.9957
Bioactivity
MY-1076 is a potent YAP inhibitor with antigastric cancer activity.MY-1076 dose-dependently induced G2/M phase block, induced YAP degradation and apoptosis, and inhibited microtubule protein polymerization.MY-1076 inhibited the proliferation of MGC-803, SGC-7901, HCT-116, and KYSE450 cells.
Smiles
OC1=C(OC)C=CC(CN(C2=CC(OC)=C(OC)C(OC)=C2)C(/C=C/C3=CC(OC)=C(OC)C(OC)=C3)=O)=C1
Molecular Formula
C29H33NO9
Molecular Weight
539.57
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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