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BRD7-IN-3

Product Specifications

Target

Epigenetic Reader Domain

Related Pathways

Chromatin/Epigenetic

Bioactivity

BRD7-IN-3 (compound 1-78) is a dual inhibitor of bromodomain-containing proteins BRD7 and BRD9, with half-maximal inhibitory concentrations (IC50s) of 1.6 μM for BRD7 and 2.7 μM for BRD9, respectively [1].

Molecular Formula

C18H18N2O2

Molecular Weight

294.35

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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