PRL 3195
Product Specifications
CAS Number
341519-04-8
Target
GPCR, Somatostatin
Related Pathways
Endocrinology/Hormones, GPCR/G Protein
Bioactivity
PRL 3195 is a somatostatin receptor antagonist with K i values of 6, 17, 66, 1000, and 1000 nM for human somatostatin receptors sst 5, sst 2, sst 3, sst 1, and sst 4, respectively [1].
Smiles
[H][C@]1(NC(=O)[C@H](CCCCN)N(C)C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccnc2)NC(=O)[C@@H](CSSC[C@H](NC1=O)C(=O)N[C@@H](Cc1ccc2ccccc2c1)C(N)=O)NC(=O)[C@@H](N)Cc1ccc(Cl)cc1)[C@@H](C)O
Molecular Formula
C58H69ClN12O9S2
Molecular Weight
1177.83
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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