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NoxaBH3

Product Specifications

Target

CXCR

Related Pathways

GPCR/G Protein|||Immunology/Inflammation|||Autophagy

Bioactivity

NoxaBH3, a cysteine-based cross-linked peptide, exhibits enhanced cell permeability and greater inhibitory efficacy against Mcl-1. It binds to the endogenous CXCR4 ligand, resulting in the formation of a ubiquitin-NoxaBH3 conjugate that is subsequently delivered to cancer cells [1].

Molecular Formula

C90H162N32O25S2

Molecular Weight

2156.68

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Product Datasheet

https://www.targetmol.com/attachment/DataSheet/64416192210665515/T76543

Available Sizes

Curated Selection

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