GR 87389
Product Specifications
CAS Number
141663-86-7
Target
Neurokinin receptor
Related Pathways
Neuroscience, GPCR/G Protein
Bioactivity
GR 87389, a potent NK2 receptor antagonist, competitively inhibits GA 64349-induced contractions in smooth muscle strips of the human detrusor, prostate, and prostatic urethra [1] [2].
Smiles
CCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H]1CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)OC(C)(C)C)C(N)=O
Molecular Formula
C47H65N9O9
Molecular Weight
900.07
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
J8009-PE 100 µL
Junctional Adhesion Molecule 1 (JAM-1, CD321, F11 Receptor, F11R, Junctional Adhesion Molecule A, JAMA, JCAM, KAT, Platelet Adhesion Molecule 1, PAM1, Platelet F11 Receptor, UNQ264/PRO301) (PE)
Sign In for Pricing
View Details 
302579-ML550 100 µL
MYCL1 (Protein L-Myc, Class E basic Helix-Loop-Helix Protein 38, bHLHe38, Protein L-Myc-1, V-myc Myelocytomatosis viral Oncogene Homolog, MYCL, BHLHE38, LMYC, MYCL1) (MaxLight 550) discontinued
Sign In for Pricing
View Details