Targefrin

Product Specifications

Target

Ephrin Receptor

Related Pathways

Tyrosine Kinase/Adaptors

Bioactivity

Targefrin is a potent antagonist targeting EphA2, exhibiting a dissociation constant of 21 nM and an IC50 value of 10.8 nM for the EphA2-LBD. It promotes receptor internalization and degradation across multiple pancreatic cancer cell lines [1].

Molecular Formula

C85H116F3N19O15

Molecular Weight

1700.94

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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